Life Science / Inhibitors/Agonists / Metabolic Enzyme / Transferase

Cat. No. Name/Description Purity
A403208 Minodronic acid monohydrate

97%
A254512 1-(2,3-Dichlorophenyl)ethanamine hydrochloride

97%
A1150708 Nevanimibe

99%
A100859 Salirasib

98%
A618355 GGTI298 Trifluoroacetate

98%
A272770 EPZ015666

98%
A645812 Perhexiline maleate

98%
A417980 Ibiglustat

98%
A711197 MAT2A inhibitor 1

98%
A1466954 FIDAS-3

95%
A1251721 K-604 2HCl

98%
A659746 4-Hydroxyphenylglyoxylate

95%
A257211 Lonafarnib

99%
A1462732 AG-270

97%
A987602 Isoastilbin

98%
A765852 GGTI-2418

98%
A412936 Tipifarnib

98%
A1258789 GDP-α-D-mannose disodium

98%
A1328405 FIDAS-5

97%
A1352619 GOT1 inhibitor-1

98%

No Data

Name/Description Transferase Other Targets Purity
Tipifarnib +++

FTase, IC50: 0.6 nM

99%+
Tolcapone +

COMT, Ki: 30 nM

99%+
Lonafarnib +++

H-ras, IC50: 1.9 nM

K-ras-4B, IC50: 2.8 nM

99%+
(E)-Daporinad ++++

NMPRTase, Ki: 0.4 nM

99%+
FTI-277 HCl ++++

FTase, IC50: 500 pM

99%+
A 922500 ++

mouse DGAT-1, IC50: 24 nM

human DGAT-1, IC50: 7 nM

99%+
Lomeguatrib ++

O6-alkylguanine-DNA-alkyltransferas, IC50: 5 nM

99%+
PF-04620110 +

DGAT1, IC50: 19 nM

98+%
LB42708 +++

FTase (K-Ras), IC50: 0.8 nM

FTase (N-ras), IC50: 1.2 nM

98%
GGTI298 Trifluoroacetate 98%+
1. Hovering the mouse over the "+" can display the specific value of the relevant IC50. The more "+", the stronger the inhibitory effect. 2. "✔" Indicates that the compound has inhibitory effects on the corresponding subtypes, but there is currently no relevant data on the intensity of inhibition.