Life Science / Inhibitors/Agonists / / Topoisomerase

Cat. No. Name/Description Purity
A191480 Valrubicin

98%
A204687 Genz-644282

99%
A1671100 Pixantrone HCl

98%
A619128 Exatecan

98%
A174646 Etoposide

98%
A257138 Temafloxacin HCl

97%
A202124 SW044248

98%
A166750 Mitoxantrone dihydrochloride

98%
A154529 Pirarubicin

98%
A122669 Topotecan HCl

98%
A910770 Exatecan Intermediate 5

98%
A182110 Isosteviol

98%
A387062 Pixantrone

98%
A207951 Mitoxantrone

98%
A783659 Nalidixic acid sodium salt

98%
A310864 Razoxane

95%
A158340 PNU-159682

98%
A472083 Amsacrine

98%
A774318 Finafloxacin hydrochloride

95%
A518842 Bisantrene

95+%

No Data

Name/Description Topo I Topo II Topo IV Topoisomerase Other Targets Purity
Ellagic acid 98%
β-Lapachone 99%+
(s)-10-hydroxycamptothecin 98+%
Camptothecin ++

Topo I, IC50: 0.68 μM

98%
Topotecan ++++

Topo I (DU-145 Luc cells), IC50: 2 nM

Topo I (MCF-7 Luc cells), IC50: 13 nM

99%+
Irinotecan HCl Trihydrate 98%
SN-38 98%
Levofloxacin hydrate 98%
Dexrazoxane 99%+
Enoxacin 99%+
Flumequine +

Topo II, IC50: 15 μM

98%
Levofloxacin 97%
Etoposide 98%
Pefloxacin mesylate dihydrate 99+%
Marbofloxacin 98+%
Voreloxin HCl 98+%
Mitoxantrone dihydrochloride PKC 98%
Nalidixic acid 98%
Novobiocin sodium 98%
Amonafide 99%+
Pirarubicin 98%+
Idarubicin HCl +++

Topo II (MCF-7 cells), IC50: 3.3 ng/mL

99%+
Teniposide 98%
Moxifloxacin 98%
Clinafloxacin 98%
Gatifloxacin 98%
Daunorubicin HCl +++

DNA synthesis, Ki: 20 nM

98%
Epirubicin HCl 99%+
1. Hovering the mouse over the "+" can display the specific value of the relevant IC50. The more "+", the stronger the inhibitory effect. 2. "✔" Indicates that the compound has inhibitory effects on the corresponding subtypes, but there is currently no relevant data on the intensity of inhibition.