Cat. No. | Name/Description | Purity |
---|---|---|
A221541 | AMI-1 free acid | 98% |
A117299 | Sorafenib Tosylate | 98% |
A662558 | Valemetostat | 99% |
A1364995 | VTP50469 | 98% |
A1867696 | BMF-219 | 98% |
A550753 | AZ505 | 99% |
A1547311 | MRTX9768 | 95% |
A713137 | Sinefungin | 98% |
A746301 | 3-Deazaneplanocin A HCl | 98% |
A345312 | EZM 2302 | 97% |
A852233 | A-395 | 98% |
A1216638 | Valemetostat tosylate | 98% |
A933282 | A-196 | 98% |
A1176455 | Onametostat | 99% |
A1327306 | MS1943 | 98% |
A211708 | UNC0379 | 98% |
A354382 | UNC0321 | 98% |
A567534 | MS049 | 98% |
A391113 | AZ505 ditrifluoroacetate | 98% |
A464128 | UNC0642 | 98% |
Name/Description | Histone Methyltransferase ↓ ↑ | Other Targets | Purity | ||||||||||||||||
---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
BRD4770 | ✔ | 99%+ | |||||||||||||||||
UNC1999 |
+++
EZH2, IC50: 2 nM EZH1, IC50: 45 nM |
99%+ | |||||||||||||||||
EPZ005687 |
++
EZH2, Ki: 24 nM |
99%+ | |||||||||||||||||
EPZ015666 |
+++
PRMT5, Ki: 5 nM |
99%+ | |||||||||||||||||
3-Deazaneplanocin A HCl |
++++
S-adenosylhomocysteine hydrolase, Ki: 50 pM |
99%+ | |||||||||||||||||
EPZ6438 |
+++
EZH2, IC50: 11 nM EZH2, Ki: 2.5 nM |
98% | |||||||||||||||||
GSK126 |
++
EZH2, IC50: 9.9 nM |
99%+ | |||||||||||||||||
MI-3 |
+
Menin-MLL, IC50: 648 nM |
98+% | |||||||||||||||||
MM-102 |
++
MLL1, IC50: 0.4 μM |
99% | |||||||||||||||||
EI1 |
++
EZH2 (Y641F), IC50: 13 nM Ezh2 (wild-type), IC50: 15 nM |
99%+ | |||||||||||||||||
SGC0946 |
++++
DOT1L, IC50: 0.3 nM |
99%+ | |||||||||||||||||
PFI-2 HCl |
++++
SETD7, Ki: 0.33 nM SETD7, IC50: 2 nM |
99%+ | |||||||||||||||||
Pinometostat |
++++
DOT1L, Ki: 80 pM |
99%+ | |||||||||||||||||
EPZ004777 |
+++
DOT1L, IC50: 0.4 nM |
99%+ | |||||||||||||||||
Entacapone |
++
COMT, IC50: 151 nM |
95% | |||||||||||||||||
UNC0379 |
+
SETD8, IC50: 7.9 μM |
99%+ | |||||||||||||||||
Menin-MLL inhibitor MI-2 |
+
Menin-MLL, IC50: 446 nM |
98+% | |||||||||||||||||
GSK343 |
+++
EZH2, IC50: 4 nM EZH1, IC50: 240 nM |
99%+ | |||||||||||||||||
BIX-01294 3HCl |
+
G9a, IC50: 2.7 μM |
99%+ | |||||||||||||||||
1. Hovering the mouse over the "+" can display the specific value of the relevant IC50. The more "+", the stronger the inhibitory effect. 2. "✔" Indicates that the compound has inhibitory effects on the corresponding subtypes, but there is currently no relevant data on the intensity of inhibition. |