Life Science / Inhibitors/Agonists / Epigenetics / Histone Demethylase

Cat. No. Name/Description Purity
A409471 GSK-J2

98%
A214803 ML324

98%
A1702949 JNJ-9350

98%
A1967108 JQKD82 trihydrochloride

98%
A1149227 Pyrene-1,6-dicarbaldehyde

95%
A608057 GSK-J4 HCl

98%
A522270 (Z)-JIB-04

97%
A1207394 Pulrodemstat benzenesulfonate

97%
A1550423 KDM2B-IN-2

98%
A1534302 PFI-90

98%
A228395 JIB-04

98%
A486013 Seclidemstat

97%
A301323 CPI-455 hydrochloride

98%
A711521 KDM4D-IN-1

98%
A1932733 AS8351

98%
A170634 IOX1

99%
A1443838 JMJD6-IN-1

98%
A114267 ORY-1001

98%
A177360 SP-2509

98+%
A1070231 SIRT2/6-IN-1

95%

No Data

Name/Description KDM1 KDM2 KDM3 KDM4 KDM5 KDM6 Other Targets Purity
OG-L002 +++

LSD1, IC50: 20 nM

99%+
ORY-1001 +++

LSD1, IC50: 20 nM

98%
SP-2509 ++++

LSD1, IC50: 13 nM

98+%
GSK2879552 2HCl +

LSD1, Ki: 1.7 μM

99%+
T-3775440 HCl ++++

LSD1, IC50: 2.1 nM

99+%
Pulrodemstat benzenesulfonate 99%+
IOX1 +

KDM2A, IC50: 1.8 μM

+++

KDM3A, IC50: 0.1 μM

++

KDM4E, IC50: 2.3 μM

KDM4C, IC50: 0.6 μM

+

KDM5C, IC50: 19 μM

+

KDM6B, IC50: 1.6 μM

99%
PFI-90 99%+
ML324 +

JMJD2, IC50: 920 nM

99%+
(Z)-JIB-04 ++

JMJD2A, IC50: 1100 nM

JMJD2E, IC50: 340 nM

++

JARID1A, IC50: 230 nM

++

JMJD3, IC50: 855 nM

97%
JIB-04 ++

JMJD2E, IC50: 435 nM

JMJD2D, IC50: 290 nM

++

JARID1A, IC50: 230 nM

++

JMJD3, IC50: 855 nM

98%
NCGC00244536 ++++

KDM4, IC50: 10 nM

95%
KDM4D-IN-1 ++

KDM4D, IC50: 0.41 μM

99%+
GSK467 ++++

KDM5B, Ki: 10 nM

99%+
GSK-J1 +++

JMJD3, IC50: 60 nM

99%+
CPI-455 ++++

KDM5A, IC50: 10 nM

++++

KDM5, IC50: 10 nM

98%
GSK-J4 HCl +++

JMJD3, IC50: 60 nM

99%+
1. Hovering the mouse over the "+" can display the specific value of the relevant IC50. The more "+", the stronger the inhibitory effect. 2. "✔" Indicates that the compound has inhibitory effects on the corresponding subtypes, but there is currently no relevant data on the intensity of inhibition.