Cat. No. | Name/Description | Purity |
---|---|---|
A409471 | GSK-J2 | 98% |
A214803 | ML324 | 98% |
A1702949 | JNJ-9350 | 98% |
A1967108 | JQKD82 trihydrochloride | 98% |
A1149227 | Pyrene-1,6-dicarbaldehyde | 95% |
A608057 | GSK-J4 HCl | 98% |
A522270 | (Z)-JIB-04 | 97% |
A1207394 | Pulrodemstat benzenesulfonate | 97% |
A1550423 | KDM2B-IN-2 | 98% |
A1534302 | PFI-90 | 98% |
A228395 | JIB-04 | 98% |
A486013 | Seclidemstat | 97% |
A301323 | CPI-455 hydrochloride | 98% |
A711521 | KDM4D-IN-1 | 98% |
A1932733 | AS8351 | 98% |
A170634 | IOX1 | 99% |
A1443838 | JMJD6-IN-1 | 98% |
A114267 | ORY-1001 | 98% |
A177360 | SP-2509 | 98+% |
A1070231 | SIRT2/6-IN-1 | 95% |
Name/Description | KDM1 ↓ ↑ | KDM2 ↓ ↑ | KDM3 ↓ ↑ | KDM4 ↓ ↑ | KDM5 ↓ ↑ | KDM6 ↓ ↑ | Other Targets | Purity | |||||||||||
---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
OG-L002 |
+++
LSD1, IC50: 20 nM |
99%+ | |||||||||||||||||
ORY-1001 |
+++
LSD1, IC50: 20 nM |
98% | |||||||||||||||||
SP-2509 |
++++
LSD1, IC50: 13 nM |
98+% | |||||||||||||||||
GSK2879552 2HCl |
+
LSD1, Ki: 1.7 μM |
99%+ | |||||||||||||||||
T-3775440 HCl |
++++
LSD1, IC50: 2.1 nM |
99+% | |||||||||||||||||
Pulrodemstat benzenesulfonate | ✔ | 99%+ | |||||||||||||||||
IOX1 |
+
KDM2A, IC50: 1.8 μM |
+++
KDM3A, IC50: 0.1 μM |
++
KDM4E, IC50: 2.3 μM KDM4C, IC50: 0.6 μM |
+
KDM5C, IC50: 19 μM |
+
KDM6B, IC50: 1.6 μM |
99% | |||||||||||||
PFI-90 | ✔ | 99%+ | |||||||||||||||||
ML324 |
+
JMJD2, IC50: 920 nM |
99%+ | |||||||||||||||||
(Z)-JIB-04 |
++
JMJD2A, IC50: 1100 nM JMJD2E, IC50: 340 nM |
++
JARID1A, IC50: 230 nM |
++
JMJD3, IC50: 855 nM |
97% | |||||||||||||||
JIB-04 |
++
JMJD2E, IC50: 435 nM JMJD2D, IC50: 290 nM |
++
JARID1A, IC50: 230 nM |
++
JMJD3, IC50: 855 nM |
98% | |||||||||||||||
NCGC00244536 |
++++
KDM4, IC50: 10 nM |
95% | |||||||||||||||||
KDM4D-IN-1 |
++
KDM4D, IC50: 0.41 μM |
99%+ | |||||||||||||||||
GSK467 |
++++
KDM5B, Ki: 10 nM |
99%+ | |||||||||||||||||
GSK-J1 |
+++
JMJD3, IC50: 60 nM |
99%+ | |||||||||||||||||
CPI-455 |
++++
KDM5A, IC50: 10 nM |
++++
KDM5, IC50: 10 nM |
98% | ||||||||||||||||
GSK-J4 HCl |
+++
JMJD3, IC50: 60 nM |
99%+ | |||||||||||||||||
1. Hovering the mouse over the "+" can display the specific value of the relevant IC50. The more "+", the stronger the inhibitory effect. 2. "✔" Indicates that the compound has inhibitory effects on the corresponding subtypes, but there is currently no relevant data on the intensity of inhibition. |