Cat. No. | Name/Description | Purity |
---|---|---|
A622861 | Emricasan | 98% |
A737788 | Arnicolide D | 97% |
A426528 | Ac-DEVD-CHO | 97% |
A230023 | Aristolactam I | 97% |
A239560 | Dehydrocorydaline chloride | 98% |
A834991 | Z-VAD-FMK | 98% |
A390989 | 5,7-Dihydroxychromone | 98% |
A100567 | VX-765 | 99% |
A149084 | Akebia saponin D | 98% |
A574284 | GRI977143 | 95% |
A169042 | Azoramide | 98% |
A131202 | PAC-1 | 98% |
A1209725 | Boc-Asp(OMe)-fluoromethyl ketone | 90% |
A724295 | 2-HBA | 98% |
A1339274 | Procaspase-3/6 activator 1 | 98+% |
A354225 | Z-VAD(OMe)-FMK | 98% |
A505764 | 5-TAMRA | 98% |
A301584 | Z-DEVD-FMK | 98% |
A553186 | Ossirene | 98% |
A173783 | Taurodeoxycholic acid sodium hydrate | 95% |
Name/Description | Capase-7 ↓ ↑ | Caspase ↓ ↑ | Caspase-1 ↓ ↑ | Caspase-10 ↓ ↑ | Caspase-2 ↓ ↑ | Caspase-3 ↓ ↑ | Caspase-4 ↓ ↑ | Caspase-5 ↓ ↑ | Caspase-6 ↓ ↑ | Caspase-8 ↓ ↑ | Caspase-9 ↓ ↑ | Other Targets | Purity | ||||||
---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Ac-DEVD-CHO |
+++
caspase-7, Ki: 1.6 nM |
+++
Caspase-1, Ki: 18 nM |
+++
caspase-10, Ki: 12 nM |
+
caspase-2, Ki: 1.71 μM |
++++
Caspase-3, Ki: 230 pM |
++
Caspase-4, Ki: 132 nM |
++
caspase-5, Ki: 205 nM |
+++
caspase-6, Ki: 31 nM |
++++
caspase-8, Ki: 0.92 nM |
++
Caspase-9, Ki: 60 nM |
99%+ | ||||||||
Emricasan | ✔ | 99%+ | |||||||||||||||||
Z-VAD(OMe)-FMK | ✔ | 99%+ | |||||||||||||||||
Z-VAD-FMK | ✔ | 99%+ | |||||||||||||||||
Z-DEVD-FMK | ✔ | 99%+ | |||||||||||||||||
VX-765 |
++++
Caspase-1, Ki: 0.8 nM |
++++
Caspase-4, Ki: <0.6 nM |
99%+ | ||||||||||||||||
Q-VD-OPh | 97% | ||||||||||||||||||
Z-IETD-FMK | ✔ | 99%+ | |||||||||||||||||
1. Hovering the mouse over the "+" can display the specific value of the relevant IC50. The more "+", the stronger the inhibitory effect. 2. "✔" Indicates that the compound has inhibitory effects on the corresponding subtypes, but there is currently no relevant data on the intensity of inhibition. |